Decitabine

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signaling-pathways

Decitabine is a clinically approved pyrimidine nucleoside analog that acts as a DNA hypomethylating (demethylating) agent, incorporating into DNA during replication and inhibiting DNA methyltransferases. It is used to reverse epigenetic silencing of genes inactivated by promoter hypermethylation, including tumor-suppressor genes silenced in cancer.

Source papers

  • Parkin activates innate immunity and promotes antitumor immune responses Michela Perego, Minjeong Yeon, Ekta Agarwal, Andrew T. Milcarek, Irene Bertolini, Chiara Camisaschi, Jagadish C. Ghosh, Hsin-Yao Tang, Nathalie Grandvaux, Marcus Ruscetti, Andrew V. Kossenkov, Sarah Preston-Alp, Italo Tempera, Noam Auslander, Dario C. Altieri · 2024 doi:10.1172/JCI180983